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Medchemexpress LLC Firazorexton hydrate (TAK-994) | 2861934-86-1 | 99.9% | 497.53 | 1 MG
Supplier: Medchemexpress LLC HY137440A1MG
Firazorexton hydrate (TAK-994) is an orally active and brain-penetrant orexin type 2 receptor (OX2R) selective agonist. It promotes wakefulness and has the potential to improve narcolepsy-like symptoms.
- Orally active and brain-penetrant orexin type 2 receptor (OX2R) selective agonist
- Promotes wakefulness
- Improves narcolepsy-like symptoms in mice models
- Increases calcium mobilization in hOX2R/CHO-K1 cells with an EC50 of 19 nM
- Activates downstream signals of OX2R
- Increases total wakefulness time in C57BL/6J mice
- Ameliorates fragmentation of wakefulness
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