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Medchemexpress LLC Fulvestrant | 129453-61-8 | 99.98% | 606.77 | 250 MG
SDP

Catalog No. 5000348787
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Fulvestrant (ICI 182780) is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC₅₀ of 9.4 nM. It also acts as a GPR30 agonist. This compound effectively inhibits the growth of ER-positive MCF-7 cells with an IC₅₀ of 0.29 nM, induces autophagy, and demonstrates antitumor efficacy. It is a potent and specific inhibitor of estrogen action, showing excellent growth-inhibitory effects in both cell and animal models of human breast cancer.

  • Pure antiestrogen
  • Potent estrogen receptor (ER) antagonist
  • GPR30 agonist
  • Inhibits growth of ER-positive MCF-7 cells
  • Induces autophagy
  • Exhibits antitumor efficacy
  • Specific inhibitor of estrogen action
  • Downregulates the estrogen receptor

Catalog No. 50-003-48787 Supplier Medchemexpress LLC Supplier No. 250MGHY13636
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Fulvestrant (ICI 182780) is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC₅₀ of 9.4 nM. It also acts as a GPR30 agonist. This compound effectively inhibits the growth of ER-positive MCF-7 cells with an IC₅₀ of 0.29 nM, induces autophagy, and demonstrates antitumor efficacy. It is a potent and specific inhibitor of estrogen action, showing excellent growth-inhibitory effects in both cell and animal models of human breast cancer.

  • Pure antiestrogen
  • Potent estrogen receptor (ER) antagonist
  • GPR30 agonist
  • Inhibits growth of ER-positive MCF-7 cells
  • Induces autophagy
  • Exhibits antitumor efficacy
  • Specific inhibitor of estrogen action
  • Downregulates the estrogen receptor

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