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Medchemexpress LLC GpTx-1 TFA | 1661050-12-9 | 99.6% | 4073.82 | 100 UG
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Supplier:  Medchemexpress LLC HYP1681A100UG

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GpTx-1 TFA is a peptide-based NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It demonstrates potent inhibitory activity against the NaV1.7 channel with an IC50 value of 10 nM. This compound also exhibits excellent selectivity for NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM).

  • Potent inhibitory activity against NaV1.7 channel with an IC50 value of 10 nM.
  • Selective for NaV1.4 (IC50 = 0.301 μM).
  • Selective for NaV1.5 (IC50 = 4.20 μM).
  • IC50 for NaV1.3 is 0.0203 μM.
  • IC50 for NaV1.8 is 12.2 μM.

Catalog No. 50-004-23669


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