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Medchemexpress LLC GpTx-1 TFA | 99.6% | 4073.82 (free base) | 1 MG
SDP

Supplier:  Medchemexpress LLC HYP1681A1MG

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GpTx-1 TFA is a peptide-based NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It demonstrates potent inhibitory activity against the NaV1.7 channel with an IC50 value of 10 nM. It also exhibits excellent selectivity for NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM), demonstrating >20-fold and >950-fold selectivity, respectively. This product is for research use only.

  • Potent inhibitory activity against NaV1.7 channel with an IC50 value of 10 nM.
  • Exhibits >20-fold selectivity for NaV1.4 (IC50 = 0.301 μM).
  • Exhibits >950-fold selectivity for NaV1.5 (IC50 = 4.20 μM).
  • Isolated from the venom of the Chilean spider Grammostola porter.

Catalog No. 50-004-23986


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