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Medchemexpress LLC GRA Ex-25 | 307983-31-9 | 99.1% | C29H36F3N3O5 | 1 ML
Supplier: Medchemexpress LLC HY5067510MM/1ML
GRA Ex-25 is an inhibitor of the glucagon receptor, with an IC50 of 56 nM for rat glucagon receptors and 55 nM for human glucagon receptors. It binds to the human glucagon receptor (h-GlucRbind) with a Ki of 63 nM and demonstrates moderate glucagon-induced adenylate cyclase inhibition (h-GlucRcyclase) with a Ki of 254 nM.
- Significantly reduces blood glucose levels in a rat model.
- Directly inhibits glucagon-stimulated hepatic glucose output.
- Suitable for research applications.
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