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Medchemexpress LLC GSK-5959 | 901245-65-6 | 99.7% | 394.47 | 10 MM 1 ML
SDP

Supplier:  Medchemexpress LLC HY1866510MM/1ML

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GSK-5959 is a potent, selective and cell permeable BRPF1 bromodomain inhibitor with an IC50 of ~80 nM.

  • Displays selectivity over the closely related family members, BRPF2 (100-fold) and BRPF3 (>1000-fold).
  • Exhibits an EC50 = 0.98 μM in cellular NanoBRET assay.
  • Has no effect on TRIM24 SUMOylation.

Catalog No. 50-003-88137


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