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Medchemexpress LLC GSK2879552 dihydrochloride | 1902123-72-1 | 99.8% | 437.40 | 100 MG
Supplier: Medchemexpress LLC HY18632A100MG
GSK2879552 dihydrochloride is an orally active, selective, and irreversible inhibitor of lysine specific demethylase 1 (LSD1/KDM1A), which has potential antineoplastic activity. For research use only, it is not sold to patients.
- Orally active.
- Selective and irreversible inhibitor of LSD1/KDM1A.
- Exhibits potential antineoplastic activity.
- Inhibits KDM1A histone demethylase activity, inducing differentiation of sorafenib-resistant cells and attenuating stemness properties in vitro.
- Depresses the transcription of Wnt antagonists and downregulates β-catenin signaling activity in sorafenib-resistant cells in vitro.
- In vivo treatment with 1.5 mg/kg exhibits tumor growth inhibition in SCLC xenograft bearing mice.
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