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Medchemexpress LLC J-2156 | 848647-56-3 | 99.9% | 468.57 | 50 MG
Supplier: Medchemexpress LLC HY11161550MG
J-2156 is a highly potent and selective somatostatin receptor type 4 (SST4 receptor) agonist, with IC50s of 0.05 nM and 0.07 nM for human and rat SST4 receptors respectively. It is used for the relief of mechanical allodynia and mechanical hyperalgesia in rat models, demonstrating nanomolar affinity for human SST4 receptors and over 400-fold subtype-selectivity against other somatostatin receptors.
- Highly potent and selective somatostatin receptor type 4 (SST4) agonist.
- Exhibits IC50s of 0.05 nM for human SST4 and 0.07 nM for rat SST4 receptors.
- Provides relief for mechanical allodynia and hyperalgesia in rats.
- Binds to human somatostatin receptor subtype 4 with a Ki of 1.2 nM.
- Offers over 400-fold subtype-selectivity against other somatostatin receptors.
- For research use only.
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