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Medchemexpress LLC Jnj-18038683 | 851376-05-1 | 99.8% | 529.97 g/mol | C26H28ClN3O7 | 10 MG
SDP

Supplier:  Medchemexpress LLC HY1988910MG

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This small-molecule research compound is a selective antagonist of the 5-hydroxytryptamine type 7 (5-HT7) receptor used in pharmacology and neuroscience studies. It shows high affinity in binding assays (pKi ≈ 8.19-8.20 for rat and human 5-HT7 in HEK293 cells), produces concentration-dependent inhibition of 5-HT-stimulated adenylyl cyclase, and alters REM sleep in rodent models. Supplied as a solid or as a DMSO solution for in vitro and in vivo research.

  • Selective 5-HT7 receptor antagonist with high binding affinity.
  • Demonstrated functional antagonism in adenylyl cyclase assays.
  • Modulates REM sleep parameters in rodent studies.
  • High purity suitable for research applications.
  • Available as solid and ready-to-use DMSO solution.
  • Store sealed and protect from moisture; follow supplier storage guidelines.

Catalog No. 50-002-99042


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