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Medchemexpress LLC L-371,257 | 162042-44-6 | 99.3% | 507.58 | 50 MG
Supplier: Medchemexpress LLC HY1501050MG
L-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective, and competitive antagonist of the oxytocin receptor. It exhibits high affinity for both the oxytocin receptor (Ki=19 nM) and the vasopressin V1a receptor (Ki=3.7 nM). This compound has been shown to stimulate weight gain in rats when administered systemically at doses of 0.5 and 1.0 mg/kg via intraperitoneal injection.
- Orally bioavailable.
- Does not penetrate the blood-brain barrier.
- Selective and competitive antagonist of the oxytocin receptor.
- High affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM).
- Stimulates weight gain in rats.
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