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Medchemexpress LLC L-745870 | 158985-00-3 | 99.9% | C18H19ClN4 | 1 ML
SDP

Catalog No. 5000354212
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L-745870 is a potent, selective, brain-penetrant, and orally active dopamine D4 receptor antagonist. It demonstrates a Ki of 0.43 nM, showing weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and moderate affinity for 5-HT2 receptors, sigma sites, and α-adrenoceptors.

  • Potent and selective dopamine D4 receptor antagonist
  • Brain-penetrant
  • Orally active
  • Exhibits weaker affinity for D2 and D3 receptors
  • Shows moderate affinity for 5-HT2 receptors, sigma sites, and α-adrenoceptors

Catalog No. 50-003-54212 Supplier Medchemexpress LLC Supplier No. HY1432510MM/1ML
May include imposed supplier surcharges.
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L-745870 is a potent, selective, brain-penetrant, and orally active dopamine D4 receptor antagonist. It demonstrates a Ki of 0.43 nM, showing weaker affinity for D2 (Ki of 960 nM) and D3 (Ki of 2300 nM) receptors, and moderate affinity for 5-HT2 receptors, sigma sites, and α-adrenoceptors.

  • Potent and selective dopamine D4 receptor antagonist
  • Brain-penetrant
  • Orally active
  • Exhibits weaker affinity for D2 and D3 receptors
  • Shows moderate affinity for 5-HT2 receptors, sigma sites, and α-adrenoceptors

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