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Medchemexpress LLC Larotinib mesylate hydrate | 2097129-93-4 | C26H36ClFN4O11S2 | 100 MG
SDP

Catalog No. 5000372921
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Larotinib mesylate hydrate is a potent, broad-spectrum, and orally active tyrosine kinase inhibitor (TKI) with EGFR as the main target with an IC50 of 0.6 nM. This compound is intended for research use only.

  • Inhibits EGFRL861Q (IC50: 0.423 nM)
  • Inhibits EGFRL858R (IC50: 0.563 nM)
  • Inhibits EGFR (WT) (IC50: 0.611 nM)
  • Inhibits EGFRT790M (IC50: 45.2 nM)
  • Inhibits HER4 (IC50: 84 nM)
  • Inhibits BLK (IC50: 102 nM)
  • Inhibits IRAK-1 (IC50: 167 nM)
  • Inhibits BTK (IC50: 196 nM)
  • Inhibits HER2 (IC50: 253 nM)

Catalog No. 50-003-72921 Supplier Medchemexpress LLC Supplier No. HY153110A100MG
May include imposed supplier surcharges.
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Larotinib mesylate hydrate is a potent, broad-spectrum, and orally active tyrosine kinase inhibitor (TKI) with EGFR as the main target with an IC50 of 0.6 nM. This compound is intended for research use only.

  • Inhibits EGFRL861Q (IC50: 0.423 nM)
  • Inhibits EGFRL858R (IC50: 0.563 nM)
  • Inhibits EGFR (WT) (IC50: 0.611 nM)
  • Inhibits EGFRT790M (IC50: 45.2 nM)
  • Inhibits HER4 (IC50: 84 nM)
  • Inhibits BLK (IC50: 102 nM)
  • Inhibits IRAK-1 (IC50: 167 nM)
  • Inhibits BTK (IC50: 196 nM)
  • Inhibits HER2 (IC50: 253 nM)

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