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TARGETMOL CHEMICALS INC MK-571 SODIUM 25MG
SDP

Supplier:  TARGETMOL CHEMICALS INC T314825MG

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Also available in 5 mg 10 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. MK-571 sodium (L-660711 sodium salt) is a selective orally active antagonist of the CysLT1 receptor. MK-571 sodium is a multidrug resistance protein-2 (ABCC2 Mrp2) inhibitor used to demonstrate the role of Mrp2 in the cellular efflux of drugs xenobiotics and their conjugates. MK-571 sodium can inhibit the synthesis of K-4′-O-GlcA (19.7 uM). MK571 dose-dependently inhibits the intracellular biosynthesis of all flavonol sulphates and glucuronides by Caco-2 cells. MK-571 sodium significantly inhibits phase-2 conjugation of kaempferol by cell-free extracts of Caco-2 and production of kaempferol-4′-O-glucuronide was competitively inhibited. In addition to inhibiting MRP2 MK571 is a potent inhibitor of enterocyte phase-2 conjugation. purity: 98%

Catalog No. 50-258-0368


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