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Medchemexpress LLC MK2-IN-3 hydrate | 1186648-22-5 | ≥99.0% | 358.39 | 10 MG
SDP

Supplier:  Medchemexpress LLC HY11245710MG

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MK2-IN-3 hydrate (compound 16) is an orally active, selective, and ATP-competitive MAPKAP-K2 (MK-2) inhibitor with an IC50 of 8.5 nM. It exhibits exceptional selectivity against MK-3 (IC50=0.21 μM), MK-5 (IC50=0.081 μM), ERK2 (IC50=3.44 μM), MNK1(IC50=5.7 μM), as well as CDK2, JNK2, IKK2, MSK1, and MSK2. It suppresses TNFα production in U397 cells with an IC50 of 4.4 μM.

  • Orally active.
  • Selective and ATP-competitive MAPKAP-K2 (MK-2) inhibitor.
  • Exceptional selectivity against MK-3, MK-5, ERK2, MNK1, CDK2, JNK2, IKK2, MSK1, and MSK2.
  • Suppresses TNFα production in U397 cells with an IC50 of 4.4 μM.

Catalog No. 50-004-38691


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