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Medchemexpress LLC Molibresib | 1260907-17-2 | 200 MG

Supplier: Medchemexpress LLC HY13032200MG
Molibresib (I-BET762; GSK525762) is a BET bromodomain inhibitor with an IC₅₀ of 32.5-42.5 nM. It binds to the tandem bromodomains of BET with high affinity and displaces a tetra-acetylated H4 peptide. It has high affinity for the BD1/BD2 domain of BRD2/3/4 proteins and inhibits OPM-2 cell proliferation.
- BET bromodomain inhibitor
- High affinity for BD1/BD2 domain of BRD2/3/4 proteins
- Inhibits OPM-2 cell proliferation
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