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Medchemexpress LLC MRS2500 tetraammonium | 630103-23-0 | 99.9% | 629.28 | 1 ML

Supplier: Medchemexpress LLC HY1086582MG
MRS2500 tetraammonium is a potent, selective, and stable antagonist of the P2Y1 receptor (Ki=0.78 nM for recombinant human P2Y1 receptor). It inhibits the ADP-induced aggregation of human platelets with an IC50 value of 0.95 nM, demonstrating antithrombotic activity.
- Potent, selective, and stable antagonist of the P2Y1 receptor.
- Inhibits ADP-induced aggregation of human platelets with an IC50 of 0.95 nM.
- Exhibits antithrombotic activity.
- Decreases acute systemic thromboembolism through selective inhibition of the P2Y1 receptor.
- Showed strong antithrombotic efficacy in preventing arterial thrombosis in the monkey ECAT model.
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