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Medchemexpress LLC MTX-531 | 2791417-66-6 | 99.9% | 453.94 | 5 MG
Supplier: Medchemexpress LLC HY1627135MG
MTX-531 is an oral drug that inhibits EGFR and PI3K isoforms (PI3Kα, PI3Kβ, PI3Kγ, and PI3Kδ). It has anti-tumor effects and acts as a weak agonist of PPARγ, which helps mitigate hyperglycemia often induced by PI3K inhibitors. It shows excellent tolerance in mice and has demonstrated concentration-dependent inhibitory effects on EGFR, P13K, and mTOR in CAL-33 cells.
- Inhibits EGFR and PI3K isoforms
- Acts as a weak agonist of PPARγ, alleviating PI3K inhibitor-induced hyperglycemia
- Demonstrates anti-tumor activity in various models
- Administered orally
- Shows excellent tolerance in mice
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