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Medchemexpress LLC N-(5-((3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl)amino)-2-methylphenyl)propionamide | 2470424-39-4 | >98.0% | 375.44 g·mol⁻¹ | C20H21N7O | 5 MG
SDP

Catalog No. 5000221059
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SGC-CK2-1 is a selective, ATP-competitive chemical probe for casein kinase 2 (CK2) with low-nanomolar enzymatic potency and demonstrated cellular activity, used for target validation and mechanistic studies in kinase research.

  • Potent enzymatic inhibition with CK2α IC50 ≈ 4.2 nM and CK2α' IC50 ≈ 2.3 nM.
  • Cell-active with nanoBRET cellular IC50s in the tens of nanomolar range.
  • High selectivity across kinases as shown by comprehensive kinome profiling.
  • Molecular weight 375.44 g·mol⁻¹ and formula C20H21N7O.
  • Soluble up to 10 mM in DMSO; DMSO stock solutions are stable at -20 °C.
  • Suitable for biochemical assays and cellular target-validation studies.

Catalog No. 50-002-21059 Supplier Medchemexpress LLC Supplier No. HY1390045MG
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SGC-CK2-1 is a selective, ATP-competitive chemical probe for casein kinase 2 (CK2) with low-nanomolar enzymatic potency and demonstrated cellular activity, used for target validation and mechanistic studies in kinase research.

  • Potent enzymatic inhibition with CK2α IC50 ≈ 4.2 nM and CK2α' IC50 ≈ 2.3 nM.
  • Cell-active with nanoBRET cellular IC50s in the tens of nanomolar range.
  • High selectivity across kinases as shown by comprehensive kinome profiling.
  • Molecular weight 375.44 g·mol⁻¹ and formula C20H21N7O.
  • Soluble up to 10 mM in DMSO; DMSO stock solutions are stable at -20 °C.
  • Suitable for biochemical assays and cellular target-validation studies.

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