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Cayman Chemical NaltrIbenmesylate 10mg
Supplier: Cayman Chemical 3897910 MG
A δ2-opioid receptor inverse agonist (Ki = 0.013 nM in CHO-DG44 cells expressing the mouse receptor); selective for δ2-opioid receptors over κ- and μ-opioid receptors (Kis = 13 and 12 nM in PC12 and COS-7 cells expressing the mouse and rat receptors, respectively); induces axonal retraction in primary mouse hippocampal neurons under both normoxic and hypoxic conditions at 1 and 10 µM; an activator of TRPM7; induces calcium influx in HEK293 cells expressing mouse TRPM7 (EC50 = 20.7 µM); reduces self-administration of alcohol or alcohol mixed with saccharin or quinine in alcohol-preferring rats at 6 mg/kg
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