Learn More
Medchemexpress LLC OARV-771 | 2683008-37-7 | 98.8% | C49H59ClN8O8S2 | 10MG

Supplier: Medchemexpress LLC HY14526410MG
OARV-771 is a VHL-based BET degrader (PROTAC) that induces proteasomal degradation of BET family proteins BRD2, BRD3, and BRD4. It demonstrates low-nanomolar degradation potency in cellular assays and is supplied as a solid with high chemical purity for research use.
- Low-nanomolar degradation potency (DC50: Brd2 ~1 nM, Brd3 ~4 nM, Brd4 ~6 nM).
- VHL-based PROTAC mechanism for targeted protein degradation.
- Improved cell permeability for cellular studies.
- High chemical purity suitable for biochemical and cell-based assays.
- Solid form for convenient handling and formulation.
- Recommended sealed cold storage to maintain stability.
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.