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Medchemexpress LLC Opiranserin hydrochloride | 1440796-75-7 | 99.6% | 430.97 | 100 MG
SDP

Supplier:  Medchemexpress LLC HY109067A50MG

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Opiranserin (VVZ-149) hydrochloride is a non-opioid and non-NSAID analgesic candidate. It functions as a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50 values of 0.86 μM and 1.3 μM, respectively. Additionally, Opiranserin hydrochloride demonstrates antagonistic activity on rP2X3 with an IC50 of 0.87 μM. It is being developed as an injectable agent for the treatment of postoperative pain. The product is intended for research use only.

  • Non-opioid and non-NSAID analgesic candidate.
  • Dual antagonist of Glycine Transporter Type 2 (GlyT2) and Serotonin Receptor 2A (5HT2A).
  • Antagonistic activity on rP2X3.
  • Development as an injectable agent for postoperative pain treatment.
  • Purity: 99.62%.

Catalog No. 50-003-44710


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