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Medchemexpress LLC Pd-168077 maleate | 630117-19-0 | 99.6% | 450.49 | 1 ML
SDP

Supplier:  Medchemexpress LLC HY21098A10MM/1ML

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PD-168077 maleate is a selective dopamine D4 receptor agonist with a Ki of 9 nM. It is intended for research use only. It exhibits intrinsic activity at the D4 receptor, leading to quinpirole-like inhibition of forskolin-stimulated cAMP accumulation or stimulation of [3H]thymidine uptake.

  • Shows >100-fold selectivity over other D2-like receptor family members and D1-like counterparts.
  • Demonstrates 20-fold selectivity over α1 and α2 receptors.
  • Exhibits 45-fold selectivity over 5-HT1A.
  • Shows 460-fold selectivity over 5-HT2A receptors.
  • Induces synaptic translocation of Ca2+/calmodulin-dependent protein kinase II in cultured prefrontal cortical neurons.

Catalog No. 50-004-00924


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