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Medchemexpress LLC PD-168077 maleate | 630117-19-0 | 99.6% | 450.49 | 50 MG
Supplier: Medchemexpress LLC HY21098A50MG
PD-168077 maleate is a selective dopamine D4 receptor agonist with a Ki of 9 nM. It exhibits high selectivity over other D2-like and D1-like receptor family members, as well as α1, α2, 5-HT1A, and 5-HT2A receptors. This compound shows intrinsic activity at the D4 receptor, inhibiting forskolin-stimulated cAMP accumulation or stimulating [3H]thymidine uptake in CHO cells expressing the human D4 receptor. In vivo, PD-168077 dose-dependently induces locomotion.
- Selective dopamine D4 receptor agonist
- Exhibits high selectivity over other D2-like, D1-like, α1, α2, 5-HT1A, and 5-HT2A receptors
- Shows intrinsic activity at the D4 receptor
- Induces locomotion in vivo
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