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Medchemexpress LLC Protac BET degrader-10 | 1957234-97-7 | 99.4% | 783.29 g/mol | C39H39ClN8O6S | 5 MG
Supplier: Medchemexpress LLC HY1127185MG
PROTAC BET Degrader-10 is a small-molecule proteolysis-targeting chimera designed to induce degradation of BET family proteins, primarily BRD4. Reported in patent WO2017007612A1 (example 37), the compound links cereblon and BRD4 ligands and has a reported DC50 of 49 nM. Typical analytical data include CAS 1957234-97-7, molecular formula C39H39ClN8O6S, molecular weight 783.29 g/mol, and purity ~99.39%.
- Induces selective BRD4 degradation in cellular assays.
- Reported DC50 of approximately 49 nM for BRD4 degradation.
- Available as solid and as a 10 mM solution in DMSO for assay flexibility.
- High chemical purity suitable for biochemical and cellular studies.
- Applicable to PROTAC mechanism-of-action and epigenetic research.
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