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Medchemexpress LLC PSB-0739 | 1052087-90-7 | 98.0% | 609.54 | 50 MG
SDP

Supplier:  Medchemexpress LLC HY108660100MG

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PSB-0739 is a high-affinity, potent, competitive, and nonselective antagonist for the platelet P2Y12 receptor, with a Ki value of 24.9 nM. This receptor is critical for platelet aggregation, and PSB-0739 demonstrates an antithrombotic effect. It is intended for research use only and not for patient treatment.

  • High-affinity potent, competitive, nonselective platelet P2Y12 receptor antagonist
  • Ki value of 24.9 nM
  • Plays a crucial role in inhibiting platelet aggregation
  • Exhibits antithrombotic effect
  • Inhibits ADP-evoked Ca2+ responses with an EC50 of 5.4±1.8 μM in THP-1 cells
  • Causes a rightward parallel shift in the ADP concentration-response curve in THP-1 cells
  • Dose-dependent and significant antihyperalgesic effect in male Wistar rats, with a minimal effective dose (mED) of 0.1 mg/kg

Catalog No. 50-003-44599


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