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Medchemexpress LLC Pulrodemstat benzenesulfonate | 2097523-60-7 | 99.6% | 10 MG
Supplier: Medchemexpress LLC HY129388B10MG
Pulrodemstat benzenesulfonate (CC-90011) is a potent, selective, reversible, and orally active inhibitor of lysine specific demethylase-1 (LSD1) with an IC50 of 0.25 nM. It exhibits less enzymatic inhibition against LSD2, MAO-A, and MAO-B. This compound induces differentiation in acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cells and demonstrates potent anticancer activity.
- Potent, selective, reversible, and orally active LSD1 inhibitor
- IC50 of 0.25 nM for LSD1
- Induces acute myeloid leukemia (AML) and small cell lung cancer (SCLC) cell differentiation
- Potent anticancer activity
- Less enzymatic inhibition against LSD2, MAO-A, and MAO-B
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