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Medchemexpress LLC Pyrrolo[3,4-b]pyrrole-5(1H)-carboxamide, N-[4-[(3-ethynylphenyl)amino]-7-methoxy-6-quinazolinyl] | 1353644-70-8 | 99.7% | 442.51 g/mol | C25H26N6O2 | 25 MG
SDP

Supplier:  Medchemexpress LLC HY10406625MG

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Theliatinib is a potent, ATP-competitive, orally active, and highly selective epidermal growth factor receptor (EGFR) inhibitor supplied as a research chemical for biochemical and cellular studies. It shows low-nanomolar potency against wild-type EGFR and measurable activity against clinically relevant mutant forms.

  • Potent, ATP-competitive EGFR inhibitor with Ki = 0.05 nM and IC50 = 3 nM.
  • Active against EGFR T790M/L858R mutant (IC50 ≈ 22 nM).
  • High purity (~99.7%) suitable for biochemical and cellular assays.
  • Molecular weight 442.51 g/mol; formula C25H26N6O2.
  • Soluble in DMSO and supplied for laboratory research use only.

Catalog No. 50-002-43800


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