Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
Learn More
Medchemexpress LLC (R)-Terazosin | 109351-34-0 | 99.76% | 50 MG
Supplier: Medchemexpress LLC HYB0371B50MG
(R)-Terazosin is an active R-enantiomer of Terazosin, functioning as a potent α1-adrenoceptor antagonist. It exhibits high affinity for α1a, α1b, and α1d-adrenoceptors, with Ki values of 6.51 nM, 1.01 nM, and 1.97 nM respectively, while showing low affinity for α2a, α2B, and α2c-adrenoceptors. This compound serves as a valuable probe for studying the functional role of adrenoceptor subtypes in various tissues and can differentiate between pharmacological effects mediated by α2-adrenoceptor subtypes in animal studies due to its weaker antagonism at α2B sites compared to its enantiomer.
- Potent α1-adrenoceptor antagonist
- Low affinity for α2a, α2B, and α2c-adrenoceptors
- Useful probe for understanding adrenoceptor subtypes and their functional roles
- Aids differentiation of pharmacological effects mediated by α2-adrenoceptor subtypes in animal studies
Product Title
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.
Spot an opportunity for improvement?