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Medchemexpress LLC (Rac)-5-Hydroxymethyl Tolterodine | 200801-70-3 | 99.05% | C22H31NO2 | 1 G
SDP

Supplier:  Medchemexpress LLC HY765701G

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(Rac)-5-Hydroxymethyl Tolterodine, an active metabolite of Tolterodine, acts as a muscarinic acetylcholine receptor (mAChR) antagonist. It exhibits Ki values ranging from 2.3 nM to 2.9 nM for M1-M5 receptors and is used in overactive bladder research.

  • Competitively inhibits carbachol-induced contraction in guinea-pig isolated urinary bladder strips (KB of 0.84 nM; pA2 of 9.14).
  • Shows significant binding to muscarinic receptors in most tissues (in vivo), with prolonged bladder duration.
  • Targets mAChR1, mAChR3, mAChR4, mAChR5.
  • Soluble in DMSO (100 mg/mL) and various aqueous/oil-based solutions (≥ 2.5 mg/mL).

Catalog No. 50-004-34020


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