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Medchemexpress LLC RN-1665 | 1803003-65-7 | 99.93% | 513.54 | 100 MG

Supplier: Medchemexpress LLC HY160900100MG
RN-1665 is an orally active TRPV4 antagonist that exhibits excellent selectivity for related TRP receptors such as TRPV1, TRPV3, and TRPM8. It serves as a TRPV4 probe for focused screens, showing IC50s of 0.26 μM for human TRPV4 and 0.39 μM for rat TRPV4.
- Orally active.
- TRPV4 antagonist.
- Exhibits excellent selectivity for related TRP receptors such as TRPV1, TRPV3, and TRPM8.
- Functions as a TRPV4 probe for focus screens.
- Has an IC50 of 0.26 μM for human TRPV4.
- Has an IC50 of 0.39 μM for rat TRPV4.
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