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Medchemexpress LLC RS-127445 | 199864-87-4 | C17H16FN3 | 1 ML
Supplier: Medchemexpress LLC HY15419A10MM/1ML
RS-127445 is a selective, high affinity, and orally bioavailable 5-HT2B receptor antagonist. It demonstrates a pKi of 9.5 and exhibits over 1000-fold selectivity for this receptor compared to numerous other receptor and ion channel binding sites.
- Selective 5-HT2B receptor antagonist
- High affinity (pKi of 9.5)
- Orally bioavailable
- Over 1000-fold selectivity compared to other receptors
- Potently blocks 5-HT evoked increases in intracellular calcium concentrations
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