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Medchemexpress LLC RS-127445 | 199864-87-4 | C17H16FN3 | 25 MG
Supplier: Medchemexpress LLC 25MGHY15419A
RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. It exhibits 1000-fold selectivity for this receptor compared to numerous other receptor and ion channel binding sites.
- Selective and high affinity 5-HT2B receptor antagonist
- Orally bioavailable
- 1000-fold selectivity compared to other receptor and ion channel binding sites
- Potently displaces [3H]-5-HT from human recombinant 5-HT2B receptors
- Blocks 5-HT-evoked increases in intracellular calcium concentrations
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