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Medchemexpress LLC RS-127445 | 199864-87-4 | C17H16FN3 | 25 MG
SDP

Catalog No. 5000375026
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RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. It exhibits 1000-fold selectivity for this receptor compared to numerous other receptor and ion channel binding sites.

  • Selective and high affinity 5-HT2B receptor antagonist
  • Orally bioavailable
  • 1000-fold selectivity compared to other receptor and ion channel binding sites
  • Potently displaces [3H]-5-HT from human recombinant 5-HT2B receptors
  • Blocks 5-HT-evoked increases in intracellular calcium concentrations

Catalog No. 50-003-75026 Supplier Medchemexpress LLC Supplier No. 25MGHY15419A
May include imposed supplier surcharges.
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RS-127445 is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist with a pKi of 9.5. It exhibits 1000-fold selectivity for this receptor compared to numerous other receptor and ion channel binding sites.

  • Selective and high affinity 5-HT2B receptor antagonist
  • Orally bioavailable
  • 1000-fold selectivity compared to other receptor and ion channel binding sites
  • Potently displaces [3H]-5-HT from human recombinant 5-HT2B receptors
  • Blocks 5-HT-evoked increases in intracellular calcium concentrations

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