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Medchemexpress LLC RS-127445 | 199864-87-4 | C17H16FN3 | 5 MG
SDP

Supplier:  Medchemexpress LLC HY15419A5MG

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This compound is a selective, high-affinity, and orally bioavailable antagonist of the 5-HT2B receptor, exhibiting a pKi of 9.5. It demonstrates significantly higher selectivity (1000-fold) for this receptor compared to numerous other receptor and ion channel binding sites.

  • High affinity for the target receptor.
  • Orally bioavailable.
  • Shows high selectivity, reducing off-target effects.
  • Effective in inhibiting serotonin-induced intracellular calcium increases.
  • Proven antagonist activity in cellular assays.

Catalog No. 50-003-76355


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