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Medchemexpress LLC SBI-810 (hydrochloride) | 2772746-58-2 | 99.6% | 483.05 | 1 ML
Supplier: Medchemexpress LLC HY164795A10MM/1ML
SBI-810 hydrochloride is a functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator. It modulates NTSR1 G protein signaling in a G protein-specific manner in the presence of the endogenous ligand, neurotensin (NT). This compound fully antagonizes NT-induced activation of Gq, partially antagonizes NT-induced activation of Gi1, and is permissive of NTSR1 activation of GoA and G12.
- Functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator.
- Modulates NTSR1 G protein signaling in a G protein-specific manner with neurotensin (NT).
- Fully antagonizes NT-induced activation of Gq.
- Partially antagonizes NT-induced activation of Gi1.
- Permissive of NTSR1 activation of GoA and G12.
- For research use only.
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