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Medchemexpress LLC SBI-810 (hydrochloride) | 2772746-58-2 | 99.6% | 483.05 | 1 ML
SDP

Catalog No. 5000391749
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SBI-810 hydrochloride is a functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator. It modulates NTSR1 G protein signaling in a G protein-specific manner in the presence of the endogenous ligand, neurotensin (NT). This compound fully antagonizes NT-induced activation of Gq, partially antagonizes NT-induced activation of Gi1, and is permissive of NTSR1 activation of GoA and G12.

  • Functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator.
  • Modulates NTSR1 G protein signaling in a G protein-specific manner with neurotensin (NT).
  • Fully antagonizes NT-induced activation of Gq.
  • Partially antagonizes NT-induced activation of Gi1.
  • Permissive of NTSR1 activation of GoA and G12.
  • For research use only.

Catalog No. 50-003-91749 Supplier Medchemexpress LLC Supplier No. HY164795A10MM/1ML
May include imposed supplier surcharges.
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SBI-810 hydrochloride is a functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator. It modulates NTSR1 G protein signaling in a G protein-specific manner in the presence of the endogenous ligand, neurotensin (NT). This compound fully antagonizes NT-induced activation of Gq, partially antagonizes NT-induced activation of Gi1, and is permissive of NTSR1 activation of GoA and G12.

  • Functionally selected β-arrestin-biased neurotensin receptor 1 (NTSR1) allosteric modulator.
  • Modulates NTSR1 G protein signaling in a G protein-specific manner with neurotensin (NT).
  • Fully antagonizes NT-induced activation of Gq.
  • Partially antagonizes NT-induced activation of Gi1.
  • Permissive of NTSR1 activation of GoA and G12.
  • For research use only.

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