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Medchemexpress LLC Siramesine (hydrochloride) | 224177-60-0 | 99.3% | C30H32ClFN2O | 100 MG
SDP

Supplier:  Medchemexpress LLC HY14221A100MG

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Siramesine hydrochloride (Lu 28-179) is a potent sigma-2 receptor agonist with subnanomolar affinity (IC50=0.12 nM) and 140-fold selectivity for sigma-2 receptors over sigma-1 receptors (IC50=17 nM). It induces cell death by destabilizing mitochondria and exhibits anti-cancer activity.

  • Potent sigma-2 receptor agonist
  • Displays subnanomolar affinity for sigma-2 receptors
  • Induces cell death by destabilizing mitochondria
  • Exhibits anti-cancer activity
  • Activates caspases in HaCaT and U-87MG cells

Catalog No. 50-003-56907


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