Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. 5000402111

Medchemexpress LLC STO-609 | 52029-86-4 | 98.2% | 314.29 | 1 ML
SDP

Supplier:  Medchemexpress LLC HY1980510MM/1ML

Encompass_Preferred

STO-609 is a selective and cell-permeable inhibitor of Ca2+/calmodulin-dependent protein kinase kinase (CaM-KK), exhibiting Ki values of 80 and 15 ng/mL for recombinant CaM-KKα and CaM-KKβ, respectively. It inhibits AMP-activated protein kinase kinase (AMPKK) activity in HeLa cell lysates (IC50 ~0.02 g/ml) and is highly selective for CaM-KK, with no significant effect on downstream CaM-KI and -IV. It also inhibits both constitutively active and wild-type CaM-KKα, and suppresses Ca2+-induced activation of CaM-KIV. The inhibition mechanism is ATP-competitive.

  • Selective and cell-permeable CaM-KK inhibitor.
  • Inhibits AMPKK activity.
  • High selectivity for CaM-KK.
  • Suppresses Ca2+-induced activation of CaM-KIV.
  • ATP-competitive inhibition mechanism.

Catalog No. 50-004-02111


May include imposed supplier surcharges.
Only null left
Add to Cart

Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.