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Medchemexpress LLC TAK-683 acetate | 99.9% | 1358.50 | 5 MG
Supplier: Medchemexpress LLC HYP2161B5MG
TAK-683 acetate is a potent full KISS1 receptor (KISS1R) agonist with improved metabolic stability. This nonapeptide metastin analog exhibits agonistic activities to KISS1R and can deplete GnRH in the hypothalamus, reducing plasma FSH, LH, and testosterone levels in vivo. It has potential for studying hormone-dependent prostate cancer.
- Potent full KISS1 receptor (KISS1R) agonist (IC50=170 pM)
- Improved metabolic stability
- Nonapeptide metastin analog
- Exhibits agonistic activities to KISS1R with EC50 values of 0.96 nM for human and 1.6 nM for rat
- Depletes GnRH in the hypothalamus
- Reduces plasma FSH, LH, and testosterone levels in vivo
- Potential for the study of hormone-dependent prostate cancer
- Molecular weight: 1358.50
- Target: Kisspeptin receptor
- Pathway: GPCR/G protein
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