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Medchemexpress LLC Tak1/map4k2 inhibitor 1 | 1315330-11-0 | 99.9% | C29H31F3N6O2 | 50 MG
Supplier: Medchemexpress LLC HY7725150MG
TAK1/MAP4K2 inhibitor 1 is a potent dual TGFβ-activated kinase 1 (TAK1) and mitogen-activated protein kinase kinase kinase kinase 2 (MAP4K2) inhibitor. It exhibits IC50s of 41.1 nM for TAK1 and 18.2 nM for MAP4K2.
- Potent dual inhibitor of TAK1 and MAP4K2
- IC50 of 41.1 nM for TAK1
- IC50 of 18.2 nM for MAP4K2
- Exhibits antiproliferative activity against parental mouse BaF3 cells harbouring Bcr/Abl
- Moderate terminal elimination half-life in mice
- Good solubility in DMSO
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