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Medchemexpress LLC Tucatinib hemiethanolate | 1429755-56-5 | 98.8% | 503.57 | 100 MG
Supplier: Medchemexpress LLC HY16069A100MG
Tucatinib hemiethanolate is a potent, orally active, and selective HER2 inhibitor. With an IC50 of 8 nM, it selectively targets HER2, showing approximately 500-fold selectivity over EGFR in cell-based assays. This compound is intended for research use only.
- Potent, orally active, and selective HER2 inhibitor
- Selectively inhibits receptor tyrosine kinase HER2 relative to EGFR
- Blocks proliferation and phosphorylation of HER2 and its downstream effector Akt
- Demonstrated anti-tumor activity and improved survival in animal models
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