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Medchemexpress LLC XPC-6444 | 2230144-21-3 | 98.9% | 50 MG
SDP

Supplier:  Medchemexpress LLC HY12877250MG

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XPC-6444 is a highly potent, isoform-selective, and CNS-penetrant inhibitor of NaV1.6, with an IC50 of 41 nM for hNaV1.6. It also effectively blocks NaV1.2, showing an IC50 of 125 nM. This compound exhibits anticonvulsant activity.

  • Highly potent and isoform-selective NaV1.6 inhibitor.
  • Effective in blocking NaV1.2.
  • Demonstrates anticonvulsant activity.
  • Shows good metabolic stability in human liver microsomes and hepatocytes.
  • Possesses low potential for MDR1 mediated efflux.
  • CNS-penetrant.

Catalog No. 50-003-38354


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