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Medchemexpress LLC Zeteletinib | 2216753-97-6 | 98.3% | 500.47 | 100 MG
SDP

Supplier:  Medchemexpress LLC HY139590100MG

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Zeteletinib is an orally active, selective RET kinase inhibitor with nanomolar potency against RET and over 300-fold selectivity against VEGFR2. It shows exquisite potency for the wild-type RET, RETV804M/L gatekeeper mutants, and the most common oncogenic RET mutation M918T. This compound exhibits potent antitumor activity and is intended for research use only.

  • Orally active and selective RET kinase inhibitor.
  • Nanomolar potency against RET.
  • Over 300-fold selectivity against VEGFR2.
  • Potent against wild-type RET, RETV804M/L gatekeeper mutants, and M918T oncogenic RET mutation.
  • Exhibits potent antitumor activity.

Catalog No. 50-003-51534


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