Promethazine-d4 (hydrochloride) is the deuterium labeled Promethazine hydrochloride. It is a first-generation antihistamine, a strong antagonist of the H1 receptor, and a moderate mACh receptor antagonist, with moderate affinity for 5-HT2A, 5-HT2C, D2, and α1-adrenergic receptors.
- Deuterium labeled compound
- Strong H1 receptor antagonist
- Moderate mACh receptor antagonist
- Moderate affinity for 5-HT2A, 5-HT2C, D2, and α1-adrenergic receptors
- Can be used as a tracer
- Suitable as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS