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Thienodiazepines

Organic heterocyclic compounds that consist of a thiophene ring fused to a diazepine ring.

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1

Medchemexpress LLC Olanzapine | 132539-06-1 | MFCD00078044 | 99.96% | C17H20N4S | 250 MG
SDP

Olanzapine is a selective, orally active monoaminergic antagonist with high affinity binding to serotonin H1, 5HT2A/2C, 5HT3, 5HT6, dopamine D1-4, muscarinic M1-5, and adrenergic α1 receptors. It is classified as an atypical antipsychotic.

  • Selective monoaminergic antagonist
  • High affinity binding to multiple serotonin, dopamine, muscarinic, and adrenergic receptors
  • Atypical antipsychotic

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2

Medchemexpress LLC Telenzepine dihydrochloride | 147416-96-4 | 99.6% | 5 MG
SDP

Telenzepine dihydrochloride is a selective and orally active muscarinic M1 receptor antagonist with a Ki of 0.94 nM. It inhibits gastric acid secretion and has antiulcer effects. In vitro, at submicromolar concentrations (100 nM), it abolishes responses to muscarine or the muscarinic component of acetylcholine. In vivo, intravenous administration potently inhibits gastric acid secretion in Ghosh-Schild rats and chronic fistula rats. Oral treatment shows significantly longer-duration antiulcer effects in modified Shay rats.

  • Selective muscarinic M1 receptor antagonist
  • Orally active
  • Inhibits gastric acid secretion
  • Antiulcer effects
  • Abolishes muscarinic responses at submicromolar concentrations
  • Potent inhibition of gastric acid secretion in vivo

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3

Medchemexpress LLC 10H-Thieno[3,4-b]benzodiazepin-10-one, 4,9-dihydro-3-methyl-4-[2-(4-methyl-1-piperazinyl)acetyl]-, hydrochloride (1:2) | 147416-96-4 | 99.6% | 100 MG
SDP

Telenzepine dihydrochloride is a selective and orally active muscarinic M1 receptor antagonist with a Ki of 0.94 nM. It inhibits gastric acid secretion and has antiulcer effects. It is for research use only.

  • Selective and orally active muscarinic M1 receptor antagonist with a Ki of 0.94 nM.
  • Inhibits gastric acid secretion.
  • Has antiulcer effects.

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4

Medchemexpress LLC Olanzapine-lactam (LY301664) | 221176-49-4 | 99.1% | 230.29 | 1 G
SDP

Olanzapine-lactam (LY301664) is a metabolite of Olanzapine. It is intended for research use.

  • High purity of 99.12%
  • Molecular weight: 230.29
  • Chemical formula: C12H10N2OS
  • Appearance: Solid
  • Color: Light yellow to yellow
  • Recommended storage: -20°C for powder, -80°C for stock solution
  • Soluble in DMSO (100 mg/mL)

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