Medchemexpress LLC Fustin | 20725-03-5 | 1 MG
Fustin ((±)-Fustin; 3,7,3',4'-Tetrahydroxyflavanone) is a potent amyloid β (Aβ) inhibitor. It increases acetylcholine (ACh) levels, choline acetyltransferase (ChAT) activity, and ChAT gene induced by Aβ (1-42). It also decreases acetyl cholinesterase (AChE) activity and AChE gene expression induced by Aβ (1-42). Fustin increases muscarinic M1 receptor gene expression and muscarinic M1 receptor binding activity. It can be used for Alzheimer's disease research.
- Potent amyloid β (Aβ) inhibitor.
- Increases acetylcholine (ACh) levels and choline acetyltransferase (ChAT) activity.
- Decreases acetylcholinesterase (AChE) activity.
- Enhances muscarinic M1 receptor expression and binding.
- Suitable for Alzheimer's disease research.