Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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586
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600
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586
R&D Systems™ GLPG 0187
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent αv integrin inhibitor
| Target | Integrin Receptor Inhibitors |
|---|---|
| CAS | 1320346-97-1 |
| Purity | 0.97 |
| Chemical Name or Material | 3-[[2,5-Dimethyl-6-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)-1-piperidinyl]-4-pyrimidinyl]amino]-N-[(4-methoxyphenyl)sulfonyl]-L-alanine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C29H37N7O5S |
587
R&D Systems™ R 547
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective cdk inhibitor
588
R&D Systems™ VH 032 amide-PEG1-amine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. VH 032-PEG1-amine
589
| CAS | 82034-46-6 |
|---|---|
| Molecular Formula | C24H31ClO7 |
590
R&D Systems™ NS 3728
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. VRAC blocker
| Target | Other Chloride Channel Blockers |
|---|---|
| CAS | 265646-85-3 |
| Purity | 0.98 |
| Chemical Name or Material | N-[3,5-bis(Trifluoromethyl)phenyl]-N'-[4-bromo-2-(2 H-tetrazol-5-yl)phenyl]urea |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C16H9BrF6N6O |
591
R&D Systems™ MK 2206 dihydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective allosteric Akt1, Akt2 and Akt3 inhibitor
| Target | Akt (Protein Kinase B) Inhibitors |
|---|---|
| CAS | 1032350-13-2 |
| Purity | 0.98 |
| Chemical Name or Material | 8-[4-(1-Aminocyclobutyl)phenyl]-9-phenyl-1,2,4-triazolo[3,4-f][1,6]naphthyridin-3(2H)-one dihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H21N5O.2HCl |
592
| CAS | 19685-09-7 |
|---|---|
| Molecular Formula | C20H16N2O5 |
593
R&D Systems™ MR 24
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective MST3 kinase binding inhibitor
| Target | Other Kinase Inhibitors |
|---|---|
| Purity | 0.98 |
| Chemical Name or Material | 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H29ClN6O3.3HCl |
594
R&D Systems™ Thalidomide 4'-oxyacetamide-alkylC8-amine
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal amine for onward chemistry
595
R&D Systems™ Lapatinib
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective dual ErbB2 (HER-2) and EGFR inhibitor (IC50 values are 9.8 and 10.2 nM, respectively)
| CAS | 231277-92-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[3-Chloro-4-[(3-fluorophenyl)methoxy]phenyl]-6-[5-[[[2-(methylsulfonyl)ethyl]amino]methyl]-2-furanyl]-4-quinazolinamine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C29H26ClFN4O4S |
| Formula Weight | 581.06 |
596
R&D Systems™ Janelia Fluor 526, SE
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Fluorogenic yellow dye; for SMLSM; λabsλem 526/550 nm
597
R&D Systems™ TL 0259
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Selective and highly potent Fgr and Lyn kinase inhibitor; orally bioavailable
| Purity | 98% |
|---|---|
| Chemical Name or Material | 3-[(6,7-Dimethoxy-4-quinazolinyl)oxy]-N-[4-[(4-ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-4-methylbenzamide dihydrochloride |
| Molecular Formula | C32H34F3N5O4.2HCl |
598
R&D Systems™ Conivaptan Hydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Very high affinity vasopressin V1A and V2 antagonist; orally bioavailable
| CAS | 168626-94-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-[4-[(4,5-Dihydro-2-methylimidazo[4,5-d][benzazepin-6(1H)-yl)carbonyl]phenyl-[1,1'-biphenyl]-2-carboxamide hydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C32H26N4O2.HCl |
| Formula Weight | 535.04 |
599
R&D Systems™ SGC AAK1 1
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. AAK1 and BMP2K inhibitor; activates Wnt signaling
| CAS | 2247894-32-0 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | N-(6-(3-((N,N-diethylsulfamoyl)amino)phenyl)-1H-indazol-3-yl)cyclopropanecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H25N5O3S |
| Formula Weight | 427.52 |
600
R&D Systems™ ARN 14494
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent serine palmitoyltransferase inhibitor
| Target | Other Transferase Inhibitors |
|---|---|
| CAS | 1037834-43-7 |
| Purity | 0.98 |
| Chemical Name or Material | rel-1-[1-[2-[(3 aR,6 AS)-Hexahydrocyclopenta[c]pyrrol-2(1 H)-yl]-2-oxoethyl]-4-piperidinyl]-2,3-dihydro-N-methyl-2-oxo-1 H-indole-5-carboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C24H32N4O3 |