Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,321
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1,321
Tocris Bioscience™ AM 6545
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High affinity and selective CB1 antagonist
| CAS | 1245626-05-4 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 20mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | AM 6545 |
| Recommended Storage | Store at 4°C |
| Synonym | 5-[4-(4-Cyano-1-butyn-1-yl)phenyl]-1-(2,4-dichlorophenyl)-N-(1,1-dioxido-4-thiomorpholinyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Molecular Formula | C26H23Cl2N5O3S |
| Formula Weight | 556.46 |
1,322
Tocris Bioscience™ cis-22a
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TRPV6 inhibitor
| Target | TRPV Inhibitors |
|---|---|
| CAS | 1819366-84-1 |
| Purity | 0.98 |
| Chemical Name or Material | 1-[cis-4-(3-Methylphenyl)cyclohexyl]-4-(3-pyridinyl)piperazine ditrifluoroacetate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H29N30.2 CF3CO2H |
1,324
Tocris Bioscience™ L-368,899 hydrochloride
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CAS: 160312-62-9 Molecular Formula: C26H43ClN4O5S2
| CAS | 160312-62-9 |
|---|---|
| Molecular Formula | C26H43ClN4O5S2 |
1,325
Tocris Bioscience™ E 2012
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γ-secretase modulator; Notch-sparing
| CAS | 870843-42-8 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | (3E)-1-[(1S)-1-(4-Fluorophenyl)ethyl]-3-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]methylene]-2-piperidone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H26FN3O2 |
| Formula Weight | 419.49 |
1,326
Tocris Bioscience™ Decitabine
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CAS: 2353-33-5 Molecular Formula: C9H13N3O4
| CAS | 2353-33-5 |
|---|---|
| Molecular Formula | C9H13N3O4 |
1,327
Tocris Bioscience™ Nafamostat mesylate
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CAS: 82956-11-4 Molecular Formula: C21H25N5O8S2
| CAS | 82956-11-4 |
|---|---|
| Molecular Formula | C21H25N5O8S2 |
1,328
Tocris Bioscience™ SEN 177
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Potent glutaminyl cyclase inhibitor; disrupts binding of SIRP-α to CD47
| Target | Other Transferase Inhibitors |
|---|---|
| CAS | 2117405-13-5 |
| Purity | 0.98 |
| Chemical Name or Material | 6 '-Fluoro-2-[4-(4-methyl-4 H-1,2,4-triazol-3-yl)-1-piperidinyl]-3,3 '-bipyridine |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H19FN6 |
1,329
Tocris Bioscience™ GW 280264X
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Potent ADAM10 and ADAM17 inhibitor
| Target | Synthetic Metalloprotease Inhibitors |
|---|---|
| CAS | 866924-39-2 |
| Purity | 0.98 |
| Chemical Name or Material | Phenylmethyl N-[(5 S)-5-[[(2 R,3 S)-3-(formylhydroxyamino)-2-(2-methylpropyl)-1-oxohexyl]amino]-6-oxo-6-(2-thiazolylamino)hexyl]carbamate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C28H41N5O6S |
1,330
Tocris Bioscience™ JTC 801
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CAS: 244218-51-7 Molecular Formula: C26H26ClN3O2
| CAS | 244218-51-7 |
|---|---|
| Molecular Formula | C26H26ClN3O2 |
1,331
Tocris Bioscience™ TCH-165
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Enhancer of 20S proteasome assembly and 20S-mediated protein degradation
| Target | Proteasome Modulators |
|---|---|
| CAS | 1446350-60-2 |
| Purity | 0.98 |
| Chemical Name or Material | Ethyl (4 R,5 R)-rel-1-benzyl-5-(4-(benzylamino)phenyl)-2-(4-methoxyphenyl)-4-phenyl-4,5-dihydro-1 H-imidazole-4-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C39H37N3O3 |
1,332
Tocris Bioscience™ QS 11
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CAS: 944328-88-5 Molecular Formula: C36H33N5O2
| CAS | 944328-88-5 |
|---|---|
| Molecular Formula | C36H33N5O2 |
1,333
Tocris Bioscience™ (S)-4-Carboxyphenylglycine
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CAS: 134052-73-6 Molecular Formula: C9H9NO4
| CAS | 134052-73-6 |
|---|---|
| Molecular Formula | C9H9NO4 |
1,334
Tocris Bioscience™ DL-Dithiothreitol
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CAS: 12-3-3483 Molecular Formula: C4H10O2S2
| CAS | 12-3-3483 |
|---|---|
| Molecular Formula | C4H10O2S2 |
1,335
Tocris Bioscience™ Idelalisib
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Potent PI 3-Kinase δ isoform inhibitor
| Target | PI 3-Kinase Inhibitors |
|---|---|
| CAS | 870281-82-6 |
| Purity | 98% |
| Chemical Name or Material | 5-Fluoro-3-phenyl-2-[(1 S)-1-(9 H-purin-6-ylamino)propyl]-4(3 H)-quinazolinone |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H18FN7O |