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  5. Tocris Bioscience™ AMG PERK 44

Tocris Bioscience™ AMG PERK 44
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Catalog No. 551750
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Catalog No. Quantity
55-175-0 50 mg
55-171-0 10 mg
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Catalog No. 55-175-0 Supplier Tocris Bioscience™ Supplier No. 5517/50
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Description

Potent and selective PERK inhibitor; orally bioavailable

AMG PERK 44 is a potent and selective PERK inhibitor (IC50 = 6 nM). Exhibits >160-fold selectivity for PERK over B-Raf and GCN2, as well as a panel of 387 other kinases. Orally bioavailable.

Specifications

Chemical Name or Material 4-[2-Amino-4-methyl-3-(2-methyl-6-quinolinyl)benzoyl]-1,2-dihydro-1-methyl-2,5-diphenyl-3H-pyrazol-3-one hydrochloride
CAS 1883548-84-2
Quantity 50 mg
Target PERK Inhibitors
Molecular Formula C34H28N4O2.HCl
Formula Weight 561.07
Purity >98%
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