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MilliporeSigma™ Calbiochem™ Adenosine A1 Receptor Antagonist I, DPCPX

Catalog No. 11914725MG Shop All MilliporeSigma Products
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11-914-725MG 25 mg
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Catalog No. 11-914-725MG Supplier MilliporeSigma™ Supplier No. 11914725MG
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Description

A blood-brain barrier permeable xanthine derivative that acts as a highly selective antagonist of Adenosine A1 receptor (A1R; Ki

A blood-brain barrier permeable xanthine derivative that acts as a highly selective antagonist of Adenosine A1 receptor (A1R; Ki = 3.9 nM, 130 nM, 1.0μM, 4.0μM for human A1, A2A, A2B, and A3 respectively). Exhibits about 1,000-fold higher affinity and a 30-fold greater selectivity for A1R when compared to theophylline. Shown to competitively antagonize the inhibition of adenylate cyclase activity via A1 adenosine receptors in rat fat cells and the stimulation of adenylate cyclase via A2 adenosine receptors in human platelets. Exhibits hypertensive properties.
TRUSTED_SUSTAINABILITY

Specifications

Color White
Description 99% by HPLC
Target Proteins A1
Molecular Formula C16H24N4O2
Formula Weight 304.4g/mol
Solubility DMSO
Content And Storage Protect from light
Form Solid
Quantity 25 mg
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