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Tocris Bioscience™ CINPA 1

Catalog No. 560550
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50 mg
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Catalog No. Quantity
56-055-0 50 mg
56-051-0 10 mg
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Catalog No. 56-055-0 Supplier Tocris Bioscience™ Supplier No. 5605/50
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Description

Potent CAR antagonist

CINPA 1 is a potent CAR antagonist (IC50 = 70 nM). Exhibits >90-fold selectivity for CAR over pregnane X receptor (PXR). Also selective over a panel of other nuclear receptors including FXR, LXR, PPARγ and RXR.

Specifications

Chemical Name or Material Ethyl [5-[(diethylamino)acetyl]-10,11-dihydro-5H-dibenz[b,f]azepin-3-yl]carbamate
CAS 102636-74-8
Quantity 50 mg
Target Constitutive Androstane Receptor Antagonists
Molecular Formula C23H29N3O3
Formula Weight 395.49
Purity >98%
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