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IRL-2500, Tocris Bioscience™ Available on GSA/VA Contract for Federal Government customers only.

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Quantity:
10mg
This item is not returnable. View return policy
169545-27-1
C36H35N3O4
573.693
UZDORQWMYRRLQV-JHOUSYSJSA-N
chembl72410,2s-2-2r-2-3,5-dimethylbenzoyl-methylamino-3-4-phenylphenyl propanoyl amino-3-1h-indol-3-yl propanoic acid,tocris-1838,d01ede,n-3-1,1'-biphenyl-4-yl-n-3,5-dimethylbenzoyl-n-methyl-d-alanyl-l-tryptophan,2s-2-2r-3-1,1'-biphenyl-4-yl-2-1-3,5-dimethylphenyl-n-methylformamido propanamido-3-1h-indol-3-yl propanoic acid,s-2-r-3-biphenyl-4-yl-2-3,5-dimethyl-benzoyl-methyl-amino-propionylamino-3-1h-indol-3-yl-propionic acid
5311192
(2S)-2-[[(2R)-2-[(3,5-dimethylbenzoyl)-methylamino]-3-(4-phenylphenyl)propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
CC1=CC(=CC(=C1)C(=O)N(C)C(CC2=CC=C(C=C2)C3=CC=CC=C3)C(=O)NC(CC4=CNC5=CC=CC=C54)C(=O)O)C
This item is not returnable. View return policy
169545-27-1
C36H35N3O4
573.693
UZDORQWMYRRLQV-JHOUSYSJSA-N
chembl72410,2s-2-2r-2-3,5-dimethylbenzoyl-methylamino-3-4-phenylphenyl propanoyl amino-3-1h-indol-3-yl propanoic acid,tocris-1838,d01ede,n-3-1,1'-biphenyl-4-yl-n-3,5-dimethylbenzoyl-n-methyl-d-alanyl-l-tryptophan,2s-2-2r-3-1,1'-biphenyl-4-yl-2-1-3,5-dimethylphenyl-n-methylformamido propanamido-3-1h-indol-3-yl propanoic acid,s-2-r-3-biphenyl-4-yl-2-3,5-dimethyl-benzoyl-methyl-amino-propionylamino-3-1h-indol-3-yl-propionic acid
5311192
(2S)-2-[[(2R)-2-[(3,5-dimethylbenzoyl)-methylamino]-3-(4-phenylphenyl)propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid
CC1=CC(=CC(=C1)C(=O)N(C)C(CC2=CC=C(C=C2)C3=CC=CC=C3)C(=O)NC(CC4=CNC5=CC=CC=C54)C(=O)O)C

Potent ETB antagonist

Potent endothelin receptor antagonist; shows some selectivity for ET B receptors (IC 50 values are 1.3 and 94 nM for ET B and ET A receptors respectively). Inhibits ET B receptor-mediated blood pressure increase and renal vascular resistance in rats in vivo.

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Formula Weight 573.69
Percent Purity >99%
Quantity 10mg
Chemical Name or Material IRL-2500

Recommended Storage : Desiccate at Room Temperature